Drug Metabolite
Drug metabolite results when a drug is metabolized into a modified form which continues to produce effects. Drug metabolism redox reactions such as heteroatom dealkylations, hydroxylations, heteroatom oxygenations, reductions, and dehydrogenations can yield active metabolites, and in rare cases even conjugation reactions can yield an active metabolite.
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Drug Metabolite Related Products (2022)
Related Products (2022)
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Antibodies (1)
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Related Compound Screening Libraries (1)
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N-Acetyl-S-(3,4-dihydroxybutyl)-L-cysteine
0 ImagesCat. No.: HY-W587741CAS No.: 144889-50-9Synonyms: Dihydroxybutyl mercapturic acid; DHBMAN-Acetyl-S-(3,4-dihydroxybutyl)-L-cysteine (Dihydroxybutyl mercapturic acid) is a biomarkersof 1,3-butadiene exposure. 1,3-Butadiene is a known human carcinogen present in cigarette smoke and in automobile exhaust.
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Dicyclohexylammonium 3-hydroxy-1-methylpropylmercapturic acid
0 ImagesCat. No.: HY-W587742CAS No.: 33164-70-4Dicyclohexylammonium 3-hydroxy-1-methylpropylmercapturic acid is a metabolite of Crotonaldehyde. Crotonaldehyde is an organic aldehyde, mainly used for the synthesis of plastics, drugs and fragrances, etc.
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3-Desacetyl Cefotaxime lactone (Standard)
0 ImagesCat. No.: HY-135394RCAS No.: 66340-33-83-Desacetyl Cefotaxime lactone (Standard) is the analytical standard of 3-Desacetyl Cefotaxime lactone. This product is intended for research and analytical applications. 3-Desacetyl Cefotaxime lactone is the active metabolite of Cefotaxime. Cefotaxime sodium salt is a third-generation cephalosporin antibiotic.
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2-Aminoflubendazole (Standard)
0 ImagesCat. No.: HY-133694RCAS No.: 82050-13-32-Aminoflubendazole (Standard) is the analytical standard of 2-Aminoflubendazole. This product is intended for research and analytical applications. 2-Aminoflubendazole is the metabolite of Benzimidazoles. Benzimidazoles (BZ) are a class of agents with activities against fungi, protozoa, and helminthes.
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γ-CEHC (Standard)
0 ImagesCat. No.: HY-113095RCAS No.: 178167-75-4Ftivazide (Standard) is the analytical standard of Ftivazide. This product is intended for research and analytical applications. Ftivazide has anti-tuberculosis activity.
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6-Hydroxy Chlorzoxazone (Standard)
0 ImagesCat. No.: HY-W016221RCAS No.: 1750-45-46-Hydroxy Chlorzoxazone (Standard) is the analytical standard of 6-Hydroxy Chlorzoxazone. This product is intended for research and analytical applications. 6-Hydroxy Chlorzoxazone is a metabolite of Chlorzoxazone (HY-B1462). Chlorzoxazone is a centrally acting muscle relaxant used to treat muscle spasm and the resulting pain or discomfort.
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Desacetylcefotaxime (Standard)
0 ImagesCat. No.: HY-126129RCAS No.: 66340-28-1Desacetylcefotaxime (Standard) is the analytical standard of Desacetylcefotaxime. This product is intended for research and analytical applications. Desacetylcefotaxime, the in vivo metabolite of Cefotaxime (CTX), possesses significant in vitro antimicrobial activity similar to the parent compound against a variety of aerobic and anaerobic bacteria.
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Eprinomectin B1a
0 ImagesCat. No.: HY-N8483CAS No.: 133305-88-1
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Lurasidone metabolite 14283
0 ImagesCat. No.: HY-G0001CAS No.: 186204-31-9Lurasidone metabolite 14283 is an active metabolite of lurasidone (HY-B0032A) and can be used in antipsychotic research.
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Posaconazole D-glucuronide
0 ImagesCat. No.: HY-172565Synonyms: SCH 56592 D-glucuronidePosaconazole D-glucuronide (SCH 56592 D-glucuronide) is a glucuronide metabolite of the antifungal agent Posaconazole (HY-17373). Posaconazole D-glucuronide can be formed in human liver microsomes catalyzed by UGT1A4.
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p,p'-DDD-13C12
0 ImagesCat. No.: HY-W750297CAS No.: 1571957-95-3Synonyms: 4,4'-DDD-13C12; p,p'-Dichlorodiphenyl dichloroethane-13C12p,p'-DDD-13C12 is 13C labeled p,p'-DDD. p,p'-DDD is a major metabolite of p,p'-DDT. p,p'-DDD occurs in the feces and livers of rats, that are given p,p'-DDT by stomach tube, but not of rats injected intraperitoneally with p,p'-DDT.
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1,2-Cyclohexanedicarboxylic acid mono 4-methyl-7-carboxy-heptyl ester
0 ImagesCat. No.: HY-W588198CAS No.: 1637562-51-61,2-Cyclohexanedicarboxylic Acid Mono 4-Methyl-7-carboxy-heptyl Ester is a secondary oxidized metabolite of di(isononyl) cyclohexane-1,2-dicarboxylate (DINCH) , an alternative for phthalate plasticizer.
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Rivastigmine metabolite-d6
0 ImagesCat. No.: HY-W020576SCAS No.: 1217706-31-4Synonyms: NAP 226-90-d6Rivastigmine metabolite-d6 (NAP 226-90-d6) is a deuterated form of Rivastigmine metabolite. Rivastigmine metabolite (NAP 226-90) is a metabolite produced by the hydrolysis of Rivastigmine (HY-17368). Rivastigmine metabolite serves as a surrogate marker to track the bioavailability, metabolic extent, and transdermal patch delivery rate of Rivastigmine.
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Berberrubine chloride (Standard)
0 ImagesCat. No.: HY-125850RCAS No.: 15401-69-1Berberrubine (chloride) (Standard) is the analytical standard of Berberrubine (chloride). This product is intended for research and analytical applications. Berberrubine chloride is an orally active metabolite of berberine. Berberrubine chloride alleviates mucosal lesions and inflammation in mouse colitis models. Berberrubine chloride has anti-inflammatory, anti-tumor, and antiviral activities.
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1-Salicylate glucuronide
0 ImagesCat. No.: HY-W410706CAS No.: 7695-70-7
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Cotinine-d3 N-β-D-Glucuronide
0 ImagesCat. No.: HY-150159SCotinine-d3 N-β-D-Glucuronide is the deuterium labeled Cotinine N-β-D-Glucuronide (HY-W588194). Cotinine N-β-D-Glucuronide is a glucuronide conjugate of the tobacco metabolite Cotinine (HY-B1178). Cotinine N-β-D-Glucuronide is promising for research of tobacco carcinogen metabolism and cognitive function.
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γ-Linolenic acid NHS ester
0 ImagesCat. No.: HY-185226CAS No.: 216447-57-3γ-Linolenic acid NHS ester is a lipid metabolite of γ-Linolenic acid (GLA) (HY-N7140), which can serve as a synthetic intermediate or probe labeling reagent for the preparation of GLA conjugates. In practical applications, γ-Linolenic acid NHS ester can be conjugated with taxanes and polysaccharides to form dual-type conjugates for drug delivery purposes.
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5-Methoxytryptamine (Standard)
0 ImagesSynonyms: O-Methylserotonin (Standard)5-Methoxytryptamine (Standard) is the analytical standard of 5-Methoxytryptamine (HY-W015169). This product is intended for research and analytical applications. 5-Methoxytryptamine, a metabolite of Melatonin, is a nonselective 5-HT receptor agonist. 5-Methoxytryptamine has no affinity for the 5-HT3 receptor. 5-Methoxytryptamine is also a potent antioxidant and has radioprotective action.
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(Rac)-3-OH-Simvastatin
0 ImagesCat. No.: HY-187569CAS No.: 134523-09-4(Rac)-3-OH-Simvastatin is a metabolite of Simvastatin (HY-17502). Simvastatin is an orally active competitive inhibitor of HMG-CoA reductase (HMGCR) with a Ki of 0.2 nM.
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THRX-195518
0 ImagesCat. No.: HY-15852CAS No.: 909800-36-8THRX-195518 is the major metabolite of Revefenacin (HY-15851), a lung-selective and long-acting muscarinic antagonist. THRX-195518 can be utilized in research related to chronic obstructive pulmonary disease.
